2020

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1. FILIPOVA, Alzbeta - MAREK, Jan - HAVELEK, Radim - PEJCHAL, Jaroslav - JELICOVA, Marcela - CIZKOVA, Jana - MAJOROŠOVÁ, Martina - MUCKOVA, Lubica - KUCERA, Tomas - PRCHAL, Lukáš - PSOTKA, Miroslav - ŽIVNÁ, Natálie - KOUTOVÁ, Darja - SINKOROVA, Zuzana - ŘEZÁČOVÁ, Martina - TICHY, Ales. Substituted piperazines as novel potential radioprotective agents. Molecules, 2020, 25(3), Art. No. 532. DOI: 10.3390/molecules25030532. ISSN 1420-3049.

2. GÓRECKI, Lukáš - ANDRYS, Rudolf - SCHMIDT, Monika - KUCERA, Tomas - PSOTKA, Miroslav - SVOBODOVÁ, Barbora - HRABCOVA, Veronika - HEPNAROVÁ, Vendula - BZONEK, Petr - JUN, Daniel - KUCA, Kamil - KORÁBEČNÝ, Jan - MUSÍLEK, Kamil. Cysteine-Targeted insecticides against A. gambiae Acetylcholinesterase are neither selective nor reversible inhibitors. ACS Medicinal Chemistry Letters, 2020, 11(1), 65-71. DOI: 10.1021/acsmedchemlett.9b00477. ISSN 1948-5875.

3. HONEGR, Jan - JUN, Daniel - KUČA, Kamil - MAREŠOVÁ, Petra. Definition of the target population for external pacemaker as a key aspect in successful medical device HTA process. Military Medical Science Letters - Vojenské zdravotnické listy, 2020, 89(2), 99-107. DOI: 10.31482/mmsl.2020.003. ISSN 0372-7025.

4. HYMPÁNOVÁ, Michaela - KUČERA, Tomáš - BENEK, Ondřej - KORÁBEČNÝ, Jan - MAREK, Jan. Searching for new antimicrobial agents by targeting bacterial nad metabolism: evaluation of frentizole derivatives selected by molecular docking. Military Medical Science Letters - Vojenské zdravotnické listy, 2020, 89(2), 66-73. DOI: 10.31482/mmsl.2020.005. ISSN 0372-7025.

5. MALIŇÁK, Dávid - DOLEŽAL, Rafael - HEPNAROVÁ, Vendula - HOZOVA, Miroslava - ANDRYS, Rudolf - BZONEK, Petr - RACAKOVA, Veronika - KORÁBEČNÝ, Jan - GÓRECKI, Lukáš - MEZEIOVÁ, Eva - PSOTKA, Miroslav - JUN, Daniel - KUČA, Kamil - MUSÍLEK, Kamil. Synthesis, in vitro screening and molecular docking of isoquinolinium-5-carbaldoximes as acetylcholinesterase and butyrylcholinesterase reactivators. Journal of Enzyme Inhibition and Medicinal Chemistry, 2020, 35(1), 478-488. DOI: 10.1080/14756366.2019.1710501. ISSN 1475-6366.

6. MAREK, Jan - TICHY, Ales - HAVELEK, Radim - MAJOROŠOVÁ, Martina - FILIPOVA, Alzbeta - ANDREJSOVA, Lenka - KUCERA, Tomas - PRCHAL, Lukáš - MUCKOVA, Lubica - ŘEZÁČOVÁ, Martina - SINKOROVA, Zuzana - PEJCHAL, Jaroslav. A novel class of small molecule inhibitors with radioprotective properties. European Journal of Medicinal Chemistry, 2020, 187(February), Art. No. UNSP111606. DOI: 10.1016/j.ejmech.2019.111606. ISSN 0223-5234.

7. MARESOVA, Petra - PETER, Lukas - HONEGR, Jan - REZNY, Lukas - PENHAKER, Marek - AUGUSTYNEK, Martin - MOHELSKA, Hana - KLIMOVA, Blanka - KUCA, Kamil. Complexity stage model of the medical device development based on economic evaluation-MedDee. Sustainability, 2020, 12(5), Art. No. 1755. DOI: 10.3390/su12051755. ISSN 2071-1050.

8. NUNHART, Patrik - KONKOLOVA, Eva - JANOVEC, Ladislav - KASPARKOVA, Jana - MALINA, Jaroslav - BRABEC, Viktor - MATEJOVA, Maria - MILTAKOVA, Beata - NOVOTNY, Ladislav - PHILLIPS, Oludotun A - UDO, Edet - KOŽURKOVÁ, Mária. Antimicrobial activity and DNA/HSA interaction of fluorinated 3,6,9-trisubstituted acridines. CHEMICAL PAPERS, 2020, 74(7), 2327-2337. DOI: 10.1007/s11696-020-01079-4. ISSN 2585-7290.

9. PATOČKA, Jiří - NAVRÁTILOVÁ, Zdeňka. Cynomorium plants: bioactive compounds and pharmacologic actions. Military Medical Science Letters - Vojenské zdravotnické listy, 2020, 89(2), 90-98. DOI: 10.31482/mmsl.2020.001. ISSN 0372-7025.

10. SABOLOVÁ, Danica - KRISTIAN, Pavol - KOŽURKOVÁ, Mária. Proflavine/acriflavine derivatives with versatile biological activities. Journal of Applied Toxicology, 2020, 40(1), 64-71. DOI: 10.1002/jat.3818. ISSN 0260-437X.

11. SHARMA, Srishti - SINGH, Namrata - NEPOVIMOVA, Eugenie - KORÁBEČNÝ, Jan - KUCA, Kamil - SATNAMI, Manmohan L - GHOSH, Kallol K. Interaction of synthesized nitrogen enriched graphene quantum dots with novel anti-Alzheimer's drugs: spectroscopic insights. Journal of Biomolecular Structure and Dynamics, 2020, 38(6), 1822-1837. DOI: 10.1080/07391102.2019.1619625. ISSN 0739-1102.

12. SCHMIDT, Monika - BENEK, Ondřej - VINKLÁŘOVÁ, Lucie - HRABINOVÁ, Martina - ZEMANOVA, Lucie - CHRIBEK, Matej - KRALOVA, Vendula - HROCH, Lukas - DOLEŽAL, Rafael - LYCKA, Antonin - PRCHAL, Lukáš - JUN, Daniel - AITKEN, Laura - GUNN-MOORE, Frank - KUCA, Kamil - MUSÍLEK, Kamil. Benzothiazolyl ureas are low micromolar and uncompetitive inhibitors of 17 beta-HSD10 with implications to Alzheimer's disease treatment. International Journal of Molecular Sciences [online], 2020, 21(6), Art. No. 2059. DOI: 10.3390/ijms21062059. ISSN 1422-0067.

13. ŽĎÁROVÁ KARASOVÁ, Jana - ŠEPSOVÁ, Vendula - ANDRYS, Rudolf - LISA, Miroslav - JOŠT, Petr - MÚČKOVÁ, Ľubica - PEJCHAL, Jaroslav - HERMAN, David - JUN, Daniel - KASSA, Jiri - KUCA, Kamil. Encapsulation of oxime K027 into cucurbit[7]uril: In vivo evaluation of safety, absorption, brain distribution and reactivation effectiveness. Toxicology Letters, 2020, 320(March), 64-72. DOI: 10.1016/j.toxlet.2019.11.021. ISSN 0378-4274.